Biological Information
Background Information:
Why choose BioPrint:
The BioPrint binding panel provides broad secondary pharmacology profiling across 135 targets, with strong GPCR coverage (73 targets) and balanced representation across key safety-relevant classes, including ion channels (18), enzymes (22), kinases (8), transporters (6), nuclear receptors (6).
This diversity enables identification of off-target safety liabilities across major organ systems.
The panel is designed for programs with constrained timelines, supporting rapid hazard assessment while delivering mechanistic insight into adverse effect risks.
No. of Assays on Panel:
135
Assays on Panel:
Family
GPCR
Name
NK1 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
100
Protein
NK1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2C Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1003
Protein
5-HT2C
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NK2 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
102
Protein
NK2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Y1 Human Neuropeptide Y GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
106
Protein
Y1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MCH1 Human Melanin-Conc. Hormone GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1115
Protein
MCH1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
delta (DOP) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
114
Protein
delta (DOP)
Organism
Human
Assay Sub Type
Binding
Family
Lipid Metabolism
Name
COX1 Human Cyclooxygenase Enzymatic LeadHunter Assay - TW
Item
116030
Protein
COX1
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
mu (MOP) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
118
Protein
mu (MOP)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H2 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1208
Protein
H2
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (Non-Selective) Rat Ion Channel [3H] TCP Binding LeadHunter Assay - FR
Item
124
Protein
NMDA(PCP site)
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
alpha2A Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
13
Protein
alpha2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
131
Protein
5-HT1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D2S Human Dopamine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1322
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H3 Human Histamine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1332
Protein
H3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2B Human Serotonin GPCR [125I](±)DOI Binding Agonist Radioligand LeadHunter Assay - FR
Item
1333
Protein
5-HT2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha2B Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1344
Protein
alpha2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H4 Human Histamine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1384
Protein
H4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
UT (GPR14) Human Urotensin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1386
Protein
UT (GPR14)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Glucagon Human Glucagon GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1407
Protein
Glucagon
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT6 Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
142
Protein
5-HT6
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT7 Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
144
Protein
5-HT7
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CRF1 Human Corticotropin-Releasing Factor GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1467
Protein
CRF1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MT1 Human Melatonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1538
Protein
MT1
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
CHT1 Human Choline Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1552
Protein
CHT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
VIP1 (VPAC1) Human VIP and PACAP GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
157
Protein
VIP1 (VPAC1)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
V1A Human Vasopressin / Oxytocin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
159
Protein
V1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha2C Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
16
Protein
alpha2C
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Rat Calcium Ion Channel Binding (Verapamil Site) LeadHunter Assay - FR
Item
163
Protein
CaV1.2 (Vera. site)
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
alpha1B Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1633
Protein
alpha1B
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav2.2 (N-type) Rat Calcium Ion Channel Binding Antagonist Radioligand LeadHunter Assay - FR
Item
164
Protein
Cav2.2 (N-type)
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
SKCa (Non-Selective) Rat Potassium Ion Channel [125I] Apamin Binding LeadHunter Assay - FR
Item
167
Protein
SKCa
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
beta1 Human Adrenoceptor GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
18
Protein
beta1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
sst1 Human Somatostatin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1940
Protein
sst1
Organism
Human
Assay Sub Type
Binding
Family
Protease
Name
ACE2 Human Angiotensin-Converting Metallo Peptidase Enzymatic LeadHunter Assay - FR
Item
1954
Protein
ACE2
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
EP2 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1955
Protein
EP2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1D Rat Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1974
Protein
5-HT1D
Organism
Rattus norvegicus (Rat)
Assay Sub Type
Binding
Family
GPCR
Name
FP Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1979
Protein
FP
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta2 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
20
Protein
beta2
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
ATPase (Na+/K+) Pig Brain Enzymatic LeadHunter Assay - FR
Item
2009
Protein
Na/K ATPase
Organism
Pig
Assay Sub Type
Enzymatic
Family
PDE
Name
PDE5 (Non-Selective) Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
204
Protein
PDE5
Organism
Human
Assay Sub Type
Enzymatic
Family
NHR
Name
RARalpha Human Retinoic Acid NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
2084
Protein
RARalpha
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
APJ Human Apelin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
2154
Protein
APJ
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
IP Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
2230
Protein
IP
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha1A Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
2338
Protein
alpha1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
AT1 Human Angiotensin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
24
Protein
AT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
AT2 Human Angiotensin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
26
Protein
AT2
Organism
Human
Assay Sub Type
Binding
Family
Steroid Metabolism
Name
Xanthine Oxidase Bovine Enzymatic LeadHunter Assay - FR
Item
276
Protein
Xanthine oxidase
Organism
Bovine
Assay Sub Type
Enzymatic
Family
Ion Channel
Name
nAChR (alpha4/beta2) Human Ion Channel Binding Agonist Radioligand LeadHunter Assay - FR
Item
3029
Protein
nAChR
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (alpha1/beta2/gamma2) Human Ion Channel [3H] Muscimol Binding Agonist Radioligand LeadHunter Assay - FR
Item
3051
Protein
GABAA
Organism
Human
Assay Sub Type
Binding
Family
Nitrogen Metabolism
Name
iNOS Mouse Nitric Oxide Synthase Enzymatic LeadHunter Assay - FR
Item
3185
Protein
iNOS
Organism
Mouse
Assay Sub Type
Enzymatic
Family
GPCR
Name
B2 Human Bradykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
33
Protein
B2
Organism
Human
Assay Sub Type
Binding
Family
Protease
Name
ACE Human Angiotensin-Converting Metallo Peptidase Enzymatic LeadHunter Assay - FR
Item
3441
Protein
ACE
Organism
Human
Assay Sub Type
Enzymatic
Family
Protease
Name
HIV-1 Protease Virus Aspartic Peptidase Enzymatic LeadHunter Assay - FR
Item
346
Protein
HIV-1 protease
Organism
Virus
Assay Sub Type
Enzymatic
Family
Transmembrane (Other)
Name
sigma (Non-Selective) Human Binding Agonist Radioligand LeadHunter Assay - FR
Item
3500
Protein
Sigma1/Sigma2
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
NET Human Norepinephrine Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
355
Protein
NET
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NOP (ORL1) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
358
Protein
NOP (ORL1)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CCR2 Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
362
Protein
CCR2
Organism
Human
Assay Sub Type
Binding
Family
Enzyme
Name
Acetylcholinesterase Human Enzymatic LeadHunter Assay - FR
Item
363
Protein
AChE
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
CB2 Human Cannabinoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
37
Protein
CB2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
mGlu5 Human Glutamate (Metabotropic) GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
3844
Protein
mGlu5
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
mGlu1 Rat Glutamate (Metabotropic) GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
3845
Protein
mGlu1
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
CCK1 (CCKA) Human Cholecystokinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
39
Protein
CCK1 (CCKA)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta3 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
3963
Protein
beta3
Organism
Homo sapiens (Human)
Assay Sub Type
Binding
Family
GPCR
Name
A2A Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4
Protein
A2A
Organism
Human
Assay Sub Type
Binding
Family
PDE
Name
PDE2A1 Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
4071
Protein
PDE2A
Organism
Human
Assay Sub Type
Enzymatic
Family
PDE
Name
PDE3B Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
4073
Protein
PDE3B
Organism
Human
Assay Sub Type
Enzymatic
Family
Enzyme
Name
PDE4D2 Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
4077
Protein
PDE4D
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
CCK2 (CCKB) Human Cholecystokinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
41
Protein
CCK2 (CCKB)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
5-HT3 Human Serotonin Ion Channel Binding Antagonist Radioligand LeadHunter Assay - FR
Item
411
Protein
5-HT3A
Organism
Human
Assay Sub Type
Binding
Family
Enzyme
Name
COX2 Human Cyclooxygenase Enzymatic LeadHunter Assay - FR
Item
4186
Protein
COX2
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
MC4 Human Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
420
Protein
MC4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1B Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
4376
Protein
5-HT1B
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
SERT Human Serotonin Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
439
Protein
SERT
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D1 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
44
Protein
D1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A1 Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
442
Protein
A1
Organism
Human
Assay Sub Type
Binding
Family
Neurotransmitter Metabolism
Name
Monoamine Oxidase A (MAO-A) Rat Binding Antagonist Radioligand LeadHunter Assay - FR
Item
443
Protein
MAO-A
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
kappa (KOP) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4461
Protein
kappa (KOP)
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
LXRbeta Human Liver X Receptor-Like NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4468
Protein
LXRbeta
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MC3 Human Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
447
Protein
MC3
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (alpha1/beta2/gamma2) Human Ion Channel [3H] Flunitrazepam Binding Agonist Radioligand LeadHunter Assay - FR
Item
4518
Protein
GABAA(BZD site)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (diltiazem site) (benzothiazepines) LeadHunter Assay - FR
Item
4549
Protein
Cav1.2 (L-type)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
PAF Human Platelet-Activating Factor GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4569
Protein
PAF
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
GR Human Glucocorticoid NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
469
Protein
GR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
GABAB (B1b/B2) Human GABAB GPCR Mass Spectrometry Binding Antagonist ligand LeadHunter Assay - FR
Item
4699
Protein
GABAB (B1/B2)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Motilin Human Motilin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
470
Protein
Motilin
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CB1 Human Cannabinoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4708
Protein
CB1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
471
Protein
5-HT2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
BB3 Human Bombesin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
472
Protein
BB3
Organism
Human
Assay Sub Type
Binding
Family
PDE
Name
PDE6 (Non-Selective) Bovine Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
478
Protein
PDE6
Organism
Bovine
Assay Sub Type
Enzymatic
Family
GPCR
Name
D3 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
48
Protein
D3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
sst4 Human Somatostatin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
482
Protein
sst4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
V2 Human Vasopressin / Oxytocin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
497
Protein
V2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A2B Human Adenosine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
5
Protein
A2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT4E Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
501
Protein
5-HT4
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (Non-Selective) Rat Ion Channel Glycine (Strychnine-Insensitive) Mass Spectrometry Binding LeadHunter Assay - FR
Item
5043
Protein
NMDA(strychine-insensitive site)
Organism
Rat
Assay Sub Type
Binding
Family
Protease
Name
MMP1 Human Matrix Metallopeptidase Enzymatic LeadHunter Assay - FR
Item
510
Protein
MMP1
Organism
Human
Assay Sub Type
Enzymatic
Family
Transporter
Name
DAT Human Dopamine Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
52
Protein
DAT
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GluK2 Human Ion Channel [3H] Kainic acid Binding LeadHunter Assay - FR
Item
5379
Protein
Kainate
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
ETA Human Endothelin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
54
Protein
ETA
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
ERalpha Human Estrogen NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
5484
Protein
ERalpha
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (Dihydropyridine Site) LeadHunter Assay - FR
Item
5538
Protein
CaV1.2 (DHP site)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Sodium Channel Site2 (Non-selective) Rat Ion Channel Batrachotoxin Mass Spectrometry Binding LeadHunter Assay - FR
Item
5572
Protein
Nav1.5
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
ETB Human Endothelin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
56
Protein
ETB
Organism
Human
Assay Sub Type
Binding
Family
Kinase
Name
p38alpha (SAPK2A) Human CMGC Kinase Enzymatic Radiometric [Km ATP] LeadHunter Assay - FR
Item
5609
Protein
p38alpha (SAPK2A)
Organism
Human
Assay Sub Type
Enzymatic
Family
Kinase
Name
ZAP70 Human TK Kinase Enzymatic Radiometric [Km ATP] LeadHunter Assay - FR
Item
5614
Protein
ZAP70
Organism
Human
Assay Sub Type
Enzymatic
Family
Kinase
Name
Fyn Human TK Kinase Enzymatic Radiometric [Km ATP] LeadHunter Assay - FR
Item
5616
Protein
Fyn
Organism
Human
Assay Sub Type
Enzymatic
Family
Kinase
Name
CDK2/CyclinA Human CMGC Kinase Enzymatic Radiometric [Km ATP] LeadHunter Assay - FR
Item
5618
Protein
CDK2
Organism
Human
Assay Sub Type
Enzymatic
Family
Kinase
Name
IR (INSR) Human RTK Kinase Enzymatic Radiometric [Km ATP] SafetyScreen - FR
Item
5623
Protein
IR
Organism
Human
Assay Sub Type
Enzymatic
Family
Kinase
Name
LYN Human TK Kinase Enzymatic Radiometric [Km ATP] LeadHunter Assay - FR
Item
5627
Protein
LYN
Organism
Human
Assay Sub Type
Enzymatic
Family
Kinase
Name
Abl (ABL1) Human TK Kinase Enzymatic Radiometric [Km ATP] LeadHunter Assay - FR
Item
5630
Protein
Abl
Organism
Human
Assay Sub Type
Enzymatic
Family
Kinase
Name
ERK2 (MAPK1) Human CMGC Kinase Enzymatic Radiometric [Km ATP] LeadHunter Assay - FR
Item
5632
Protein
ERK2
Organism
Human
Assay Sub Type
Enzymatic
Family
Kinase
Name
Flt-1 (VEGFR1) (FLT1) Human RTK Kinase Enzymatic Radiometric [Km ATP] SafetyScreen - FR
Item
5641
Protein
Flt-1 (VEGFR1)
Organism
Human
Assay Sub Type
Enzymatic
Family
Kinase
Name
CaMK2alpha (CAMK2A) (Active) Human CAMK Kinase Enzymatic Radiometric [Km ATP] LeadHunter Assay - FR
Item
5642
Protein
CaMK2alpha
Organism
Human
Assay Sub Type
Enzymatic
Family
Ion Channel
Name
GABAA (alpha1/beta2/gamma2) Human Ion Channel Picrotoxinin Mass Spectrometry Binding Antagonist Ligand LeadHunter Assay - FR
Item
5666
Protein
GABAA
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
GAT1 Human GABA Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
5773
Protein
GAT-1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CysLT1 Human Leukotriene GPCR Mass Spectrometry Binding Agonist ligand LeadHunter Assay - FR
Item
5841
Protein
CYSLT1
Organism
Human
Assay Sub Type
Binding
Family
Protease
Name
MMP9 Human Matrix Metallopeptidase Enzymatic LeadHunter assay - FR
Item
5850
Protein
MMP9
Organism
Human
Assay Sub Type
Enzymatic
Family
Protease
Name
MMP2 Human Matrix Metallopeptidase Enzymatic LeadHunter assay - FR
Item
5870
Protein
MMP2
Organism
Human
Assay Sub Type
Enzymatic
Family
Ion Channel
Name
Glutamate (NMDA, NR1/NR2A) Human Ion Channel [3H] CGP-39653 Binding LeadHunter Assay - FR
Item
5875
Protein
GluN1 / GluN2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A3 Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
6
Protein
A3
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (AMPA, Non-Selective) Rat Ion Channel [3H] AMPA Binding LeadHunter Assay - FR
Item
64
Protein
AMPA
Organism
Rat
Assay Sub Type
Binding
Family
NHR
Name
PPARgamma Human NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
641
Protein
PPARgamma
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MC1 Mouse Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
644
Protein
MC1
Organism
Mouse
Assay Sub Type
Binding
Family
Protease
Name
beta-Secretase 1 Human Pepsin Aspartic Peptidase Enzymatic LeadHunter Assay - FR
Item
701
Protein
beta-Secretase 1
Organism
Human
Assay Sub Type
Enzymatic
Family
Cell Surface (Other)
Name
TNF-alpha Human Binding Agonist Radioligand LeadHunter Assay - FR
Item
76
Protein
TNF-alpha
Organism
Human
Assay Sub Type
Binding
Family
Protease
Name
Caspase 3 Human Caspase Cysteine Peptidase Enzymatic LeadHunter Assay - FR
Item
774
Protein
Caspase 3
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
H1 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
870
Protein
H1
Organism
Human
Assay Sub Type
Binding
Family
Cytosolic (Other)
Name
QR2 / MT3 Hamster Binding Agonist Radioligand LeadHunter Assay - FR
Item
88
Protein
QR2 / MT3
Organism
Hamster
Assay Sub Type
Binding
Family
GPCR
Name
M1 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
91
Protein
M1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
GHSR Human Ghrelin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
928
Protein
GHSR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M2 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
93
Protein
M2
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
AR Human Androgen NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
933
Protein
AR
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
nAChR (Alpha1, Muscle-Type) Human Ion Channel Binding Antagonist Radioligand LeadHunter Assay - FR
Item
936
Protein
nAChR-α1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M3 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
95
Protein
M3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M4 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
96
Protein
M4
Organism
Human
Assay Sub Type
Binding
Testing Information
Test Sample Requirements:
Minimum for Screen: 220 µl of 10 mM stock -OR- 1.10 mg (pre-weighed) for 10µM final testing.
(PBS or HBSS working solutions are not compatible)
Turnaround Time
Standard:
15 Business Days
Additional Information
Brand:
SafetyScreen
Testing Location:
France - Celle L'Evescault
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