Biological Information

Background Information:


Why choose BioPrint:
The BioPrint binding panel provides broad secondary pharmacology profiling across 135 targets, with strong GPCR coverage (73 targets) and balanced representation across key safety-relevant classes, including ion channels (18), enzymes (22), kinases (8), transporters (6), nuclear receptors (6).
This diversity enables identification of off-target safety liabilities across major organ systems.
The panel is designed for programs with constrained timelines, supporting rapid hazard assessment while delivering mechanistic insight into adverse effect risks.


Key Benefits from screening with BioPrint:
Cost-effective
package for screening and profiling activities.
Visualize and interpret your data with In Vitro Safety Insight: identify organ risks, rank compounds, and access follow-up assay recommendations (available in your online account).
Fast start: profiling begins the day after compound receipt. No scheduling, to meet tight deadline and ensure fast TAT.
Access data early:
results released as they are validated.
Final report
delivered electronically with notification.
Eligible for the French Crédit Impôt Recherche (CIR) tax incentive.


What’s Next after BioPrint:
Follow-up your hits with Binding or Functional IC₅₀/EC₅₀.

No. of Assays on Panel:

135

Assays on Panel:

Family

GPCR

Name

Item

100

Protein

NK1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1003

Protein

5-HT2C

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

102

Protein

NK2

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

106

Protein

Y1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1115

Protein

MCH1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

114

Protein

delta (DOP)

Organism

Human

Assay Sub Type

Binding

Family

Lipid Metabolism

Name

Item

116030

Protein

COX1

Organism

Human

Assay Sub Type

Enzymatic

Family

GPCR

Name

Item

118

Protein

mu (MOP)

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1208

Protein

H2

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

124

Protein

NMDA(PCP site)

Organism

Rat

Assay Sub Type

Binding

Family

GPCR

Name

Item

13

Protein

alpha2A

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

131

Protein

5-HT1A

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1322

Protein

D2

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1332

Protein

H3

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1333

Protein

5-HT2B

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1344

Protein

alpha2B

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1384

Protein

H4

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1386

Protein

UT (GPR14)

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1407

Protein

Glucagon

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

142

Protein

5-HT6

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

144

Protein

5-HT7

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1467

Protein

CRF1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1538

Protein

MT1

Organism

Human

Assay Sub Type

Binding

Family

Transporter

Name

Item

1552

Protein

CHT1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

157

Protein

VIP1 (VPAC1)

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

159

Protein

V1A

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

16

Protein

alpha2C

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

163

Protein

CaV1.2 (Vera. site)

Organism

Rat

Assay Sub Type

Binding

Family

GPCR

Name

Item

1633

Protein

alpha1B

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

164

Protein

Cav2.2 (N-type)

Organism

Rat

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

167

Protein

SKCa

Organism

Rat

Assay Sub Type

Binding

Family

GPCR

Name

Item

18

Protein

beta1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1940

Protein

sst1

Organism

Human

Assay Sub Type

Binding

Family

Protease

Name

Item

1954

Protein

ACE2

Organism

Human

Assay Sub Type

Enzymatic

Family

GPCR

Name

Item

1955

Protein

EP2

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

1974

Protein

5-HT1D

Organism

Rattus norvegicus (Rat)

Assay Sub Type

Binding

Family

GPCR

Name

Item

1979

Protein

FP

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

20

Protein

beta2

Organism

Human

Assay Sub Type

Binding

Family

Transporter

Name

Item

2009

Protein

Na/K ATPase

Organism

Pig

Assay Sub Type

Enzymatic

Family

PDE

Name

Item

204

Protein

PDE5

Organism

Human

Assay Sub Type

Enzymatic

Family

NHR

Name

Item

2084

Protein

RARalpha

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

2154

Protein

APJ

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

2230

Protein

IP

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

2338

Protein

alpha1A

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

24

Protein

AT1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

26

Protein

AT2

Organism

Human

Assay Sub Type

Binding

Family

Steroid Metabolism

Name

Item

276

Protein

Xanthine oxidase

Organism

Bovine

Assay Sub Type

Enzymatic

Family

Ion Channel

Name

Item

3029

Protein

nAChR

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

3051

Protein

GABAA

Organism

Human

Assay Sub Type

Binding

Family

Nitrogen Metabolism

Name

Item

3185

Protein

iNOS

Organism

Mouse

Assay Sub Type

Enzymatic

Family

GPCR

Name

Item

33

Protein

B2

Organism

Human

Assay Sub Type

Binding

Family

Protease

Name

Item

3441

Protein

ACE

Organism

Human

Assay Sub Type

Enzymatic

Family

Protease

Name

Item

346

Protein

HIV-1 protease

Organism

Virus

Assay Sub Type

Enzymatic

Family

Transmembrane (Other)

Name

Item

3500

Protein

Sigma1/Sigma2

Organism

Human

Assay Sub Type

Binding

Family

Transporter

Name

Item

355

Protein

NET

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

358

Protein

NOP (ORL1)

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

362

Protein

CCR2

Organism

Human

Assay Sub Type

Binding

Family

Enzyme

Name

Item

363

Protein

AChE

Organism

Human

Assay Sub Type

Enzymatic

Family

GPCR

Name

Item

37

Protein

CB2

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

3844

Protein

mGlu5

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

3845

Protein

mGlu1

Organism

Rat

Assay Sub Type

Binding

Family

GPCR

Name

Item

39

Protein

CCK1 (CCKA)

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

3963

Protein

beta3

Organism

Homo sapiens (Human)

Assay Sub Type

Binding

Family

GPCR

Name

Item

4

Protein

A2A

Organism

Human

Assay Sub Type

Binding

Family

PDE

Name

Item

4071

Protein

PDE2A

Organism

Human

Assay Sub Type

Enzymatic

Family

PDE

Name

Item

4073

Protein

PDE3B

Organism

Human

Assay Sub Type

Enzymatic

Family

Enzyme

Name

Item

4077

Protein

PDE4D

Organism

Human

Assay Sub Type

Enzymatic

Family

GPCR

Name

Item

41

Protein

CCK2 (CCKB)

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

411

Protein

5-HT3A

Organism

Human

Assay Sub Type

Binding

Family

Enzyme

Name

Item

4186

Protein

COX2

Organism

Human

Assay Sub Type

Enzymatic

Family

GPCR

Name

Item

420

Protein

MC4

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

4376

Protein

5-HT1B

Organism

Human

Assay Sub Type

Binding

Family

Transporter

Name

Item

439

Protein

SERT

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

44

Protein

D1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

442

Protein

A1

Organism

Human

Assay Sub Type

Binding

Family

Neurotransmitter Metabolism

Name

Item

443

Protein

MAO-A

Organism

Rat

Assay Sub Type

Binding

Family

GPCR

Name

Item

4461

Protein

kappa (KOP)

Organism

Human

Assay Sub Type

Binding

Family

NHR

Name

Item

4468

Protein

LXRbeta

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

447

Protein

MC3

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

4518

Protein

GABAA(BZD site)

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

4549

Protein

Cav1.2 (L-type)

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

4569

Protein

PAF

Organism

Human

Assay Sub Type

Binding

Family

NHR

Name

Item

469

Protein

GR

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

4699

Protein

GABAB (B1/B2)

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

470

Protein

Motilin

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

4708

Protein

CB1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

471

Protein

5-HT2A

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

472

Protein

BB3

Organism

Human

Assay Sub Type

Binding

Family

PDE

Name

Item

478

Protein

PDE6

Organism

Bovine

Assay Sub Type

Enzymatic

Family

GPCR

Name

Item

48

Protein

D3

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

482

Protein

sst4

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

497

Protein

V2

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

5

Protein

A2B

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

501

Protein

5-HT4

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

5043

Protein

NMDA(strychine-insensitive site)

Organism

Rat

Assay Sub Type

Binding

Family

Protease

Name

Item

510

Protein

MMP1

Organism

Human

Assay Sub Type

Enzymatic

Family

Transporter

Name

Item

52

Protein

DAT

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

5379

Protein

Kainate

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

54

Protein

ETA

Organism

Human

Assay Sub Type

Binding

Family

NHR

Name

Item

5484

Protein

ERalpha

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

5538

Protein

CaV1.2 (DHP site)

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

5572

Protein

Nav1.5

Organism

Rat

Assay Sub Type

Binding

Family

GPCR

Name

Item

56

Protein

ETB

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

5609

Protein

p38alpha (SAPK2A)

Organism

Human

Assay Sub Type

Enzymatic

Family

Kinase

Name

Item

5614

Protein

ZAP70

Organism

Human

Assay Sub Type

Enzymatic

Family

Kinase

Name

Item

5616

Protein

Fyn

Organism

Human

Assay Sub Type

Enzymatic

Family

Kinase

Name

Item

5618

Protein

CDK2

Organism

Human

Assay Sub Type

Enzymatic

Family

Kinase

Name

Item

5623

Protein

IR

Organism

Human

Assay Sub Type

Enzymatic

Family

Kinase

Name

Item

5627

Protein

LYN

Organism

Human

Assay Sub Type

Enzymatic

Family

Kinase

Name

Item

5630

Protein

Abl

Organism

Human

Assay Sub Type

Enzymatic

Family

Kinase

Name

Item

5632

Protein

ERK2

Organism

Human

Assay Sub Type

Enzymatic

Family

Kinase

Name

Item

5641

Protein

Flt-1 (VEGFR1)

Organism

Human

Assay Sub Type

Enzymatic

Family

Kinase

Name

Item

5642

Protein

CaMK2alpha

Organism

Human

Assay Sub Type

Enzymatic

Family

Ion Channel

Name

Item

5666

Protein

GABAA

Organism

Human

Assay Sub Type

Binding

Family

Transporter

Name

Item

5773

Protein

GAT-1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

5841

Protein

CYSLT1

Organism

Human

Assay Sub Type

Binding

Family

Protease

Name

Item

5850

Protein

MMP9

Organism

Human

Assay Sub Type

Enzymatic

Family

Protease

Name

Item

5870

Protein

MMP2

Organism

Human

Assay Sub Type

Enzymatic

Family

Ion Channel

Name

Item

5875

Protein

GluN1 / GluN2A

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

6

Protein

A3

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

64

Protein

AMPA

Organism

Rat

Assay Sub Type

Binding

Family

NHR

Name

Item

641

Protein

PPARgamma

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

644

Protein

MC1

Organism

Mouse

Assay Sub Type

Binding

Family

Protease

Name

Item

701

Protein

beta-Secretase 1

Organism

Human

Assay Sub Type

Enzymatic

Family

Cell Surface (Other)

Name

Item

76

Protein

TNF-alpha

Organism

Human

Assay Sub Type

Binding

Family

Protease

Name

Item

774

Protein

Caspase 3

Organism

Human

Assay Sub Type

Enzymatic

Family

GPCR

Name

Item

870

Protein

H1

Organism

Human

Assay Sub Type

Binding

Family

Cytosolic (Other)

Name

Item

88

Protein

QR2 / MT3

Organism

Hamster

Assay Sub Type

Binding

Family

GPCR

Name

Item

91

Protein

M1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

928

Protein

GHSR

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

93

Protein

M2

Organism

Human

Assay Sub Type

Binding

Family

NHR

Name

Item

933

Protein

AR

Organism

Human

Assay Sub Type

Binding

Family

Ion Channel

Name

Item

936

Protein

nAChR-α1

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

95

Protein

M3

Organism

Human

Assay Sub Type

Binding

Family

GPCR

Name

Item

96

Protein

M4

Organism

Human

Assay Sub Type

Binding

Testing Information

Test Sample Requirements:

Minimum for Screen: 220 µl of 10 mM stock -OR- 1.10 mg (pre-weighed) for 10µM final testing.
(PBS or HBSS working solutions are not compatible)

Turnaround Time

Standard:

15 Business Days

Additional Information

Brand:

SafetyScreen

Testing Location:

France - Celle L'Evescault

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