Biological Information

Background Information:

SH2MAX Profiling Panel is a pre-defined panel of 102 human SRC Homology 2 domain-containing wild-type and mutant targets from multiple target families including STATs, kinases, phosphatases, phospholipases, E3 ligases, adaptor proteins, GEFs, and signal regulators for convenient, rapid selectivity screening of therapeutics.

No. of Assays on Panel:

102

Assays on Panel:

Family

Nuclear Protein

Name

Item

84-0005-1001

Protein

STAT1

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1002

Protein

STAT2

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1003

Protein

STAT3

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1004

Protein

STAT4

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1005

Protein

STAT5A

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1006

Protein

STAT5B

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1007

Protein

STAT6

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1008

Protein

STAT5B

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1009

Protein

STAT3

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1010

Protein

STAT3

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1011

Protein

Abl

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1012

Protein

Arg

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1013

Protein

BLK

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1014

Protein

Brk (PTK6)

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1015

Protein

CSK

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1016

Protein

Fer

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1017

Protein

FES

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1018

Protein

FGR

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1019

Protein

FRK (PTK5)

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1020

Protein

Fyn

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1021

Protein

HCK

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1022

Protein

ITK

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1023

Protein

Lck

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1024

Protein

LYN

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1025

Protein

PIK3R1 (p85alpha)

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1026

Protein

PIK3R1 (p85alpha)

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1027

Protein

PIK3R2 (p85beta)

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1028

Protein

PIK3R2 (p85beta)

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1029

Protein

PIK3R3 (p55gamma)

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1030

Protein

PIK3R3 (p55gamma)

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1031

Protein

Src

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1032

Protein

Srm

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1033

Protein

Syk

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1034

Protein

TEC

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1035

Protein

YES

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1036

Protein

ZAP70

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1037

Protein

SH2B2

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1038

Protein

BLNK

Organism

Human

Assay Sub Type

Binding

Family

Ubiquitin Modifying

Name

Item

84-0005-1039

Protein

Cbl

Organism

Human

Assay Sub Type

Binding

Family

Ubiquitin Modifying

Name

Item

84-0005-1040

Protein

CBLB

Organism

Human

Assay Sub Type

Binding

Family

Ubiquitin Modifying

Name

Item

84-0005-1041

Protein

CBLC

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1042

Protein

CISH

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1043

Protein

CRK

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1044

Protein

CRKL

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1045

Protein

DAPP1

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1046

Protein

GRAP2

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1047

Protein

GRAP

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1048

Protein

GRB10

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1049

Protein

GRB14

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1050

Protein

GRB2

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1051

Protein

GRB7

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1052

Protein

HSH2D

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1053

Protein

SH2B3

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1054

Protein

CTK

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1055

Protein

CLNK

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1056

Protein

NCK1

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1057

Protein

NCK2

Organism

Human

Assay Sub Type

Binding

Family

Lipid Metabolism

Name

Item

84-0005-1058

Protein

PLCgamma1

Organism

Human

Assay Sub Type

Binding

Family

Lipid Metabolism

Name

Item

84-0005-1059

Protein

PLCgamma1

Organism

Human

Assay Sub Type

Binding

Family

Lipid Metabolism

Name

Item

84-0005-1060

Protein

PLCgamma2

Organism

Human

Assay Sub Type

Binding

Family

Lipid Metabolism

Name

Item

84-0005-1061

Protein

PLCgamma2

Organism

Human

Assay Sub Type

Binding

Family

Phosphatase

Name

Item

84-0005-1062

Protein

SHP2

Organism

Human

Assay Sub Type

Binding

Family

Phosphatase

Name

Item

84-0005-1063

Protein

SHP2

Organism

Human

Assay Sub Type

Binding

Family

Phosphatase

Name

Item

84-0005-1064

Protein

SHP1

Organism

Human

Assay Sub Type

Binding

Family

Phosphatase

Name

Item

84-0005-1065

Protein

SHP1

Organism

Human

Assay Sub Type

Binding

Family

Nucleotide Signaling

Name

Item

84-0005-1066

Protein

RASA1

Organism

Human

Assay Sub Type

Binding

Family

Nucleotide Signaling

Name

Item

84-0005-1067

Protein

RASA1

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1068

Protein

SH2B1

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1069

Protein

SH21A

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1070

Protein

SH21B

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1071

Protein

SH2D6

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1072

Protein

3BP2

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1073

Protein

SHB

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1074

Protein

SHC1

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1075

Protein

SHC2

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1076

Protein

SHC3

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1077

Protein

SHC4

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1078

Protein

SHF

Organism

Human

Assay Sub Type

Binding

Family

Phosphatase

Name

Item

84-0005-1079

Protein

SHIP1 (INPP5D)

Organism

Human

Assay Sub Type

Binding

Family

Phosphatase

Name

Item

84-0005-1080

Protein

SHIP2 (INPPL1)

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1081

Protein

SLAP2

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1082

Protein

LCP2

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1083

Protein

SOCS1

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1084

Protein

SOCS2

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1085

Protein

SOCS3

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1086

Protein

SOCS4

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1088

Protein

SOCS6

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1089

Protein

SOCS7

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1090

Protein

STAP1

Organism

Human

Assay Sub Type

Binding

Family

Adaptor

Name

Item

84-0005-1091

Protein

STAP2

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1092

Protein

STAT3

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1093

Protein

STAT3

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1094

Protein

STAT3

Organism

Human

Assay Sub Type

Binding

Family

Immune System

Name

Item

84-0005-1095

Protein

STAT3

Organism

Human

Assay Sub Type

Binding

Family

Cytosolic (Other)

Name

Item

84-0005-1096

Protein

TENS1

Organism

Human

Assay Sub Type

Binding

Family

Cytosolic (Other)

Name

Item

84-0005-1097

Protein

TENS2

Organism

Human

Assay Sub Type

Binding

Family

Cytosolic (Other)

Name

Item

84-0005-1098

Protein

TENS3

Organism

Human

Assay Sub Type

Binding

Family

Cytosolic (Other)

Name

Item

84-0005-1099

Protein

TENS4

Organism

Human

Assay Sub Type

Binding

Family

Kinase

Name

Item

84-0005-1100

Protein

TXK

Organism

Human

Assay Sub Type

Binding

Family

Nucleotide Signaling

Name

Item

84-0005-1101

Protein

VAV

Organism

Human

Assay Sub Type

Binding

Family

Nucleotide Signaling

Name

Item

84-0005-1102

Protein

VAV2

Organism

Human

Assay Sub Type

Binding

Family

Nucleotide Signaling

Name

Item

84-0005-1103

Protein

VAV3

Organism

Human

Assay Sub Type

Binding

Family:

Signaling Pathway

Sub Family:

SH2 Domain Containing

Organism:

Human

Assay Information

Assay Type:

Biochemical

Assay Sub Type:

Binding

Testing Information

Test Sample Requirements:

50uL of a 1000X stock based on the top or final concentration being tested

Turnaround Time

Standard:

14 Business Days

Clinical Relevance

Therapeutic Area:

Oncology/ Inflammation/ Autoimmune

Additional Information

Brand:

SH2scan - DiscoverX

Testing Location:

USA - San Diego, CA