Biological Information

Family:

Kinase

Sub Family:

CAMK

Class:

Protein Serine/Threonine

Protein Name:

AMPKalpha1

Uniprot Number:

Q13131

Protein Aliases:

AMPK, alpha, 1

Gene Name:

PRKAA1

Gene ID:

5562

Gene Aliases:

AMPKa1

Accession Number:

AF100763 (a1)/NM_006

Organism:

Human

Assay Information

Assay Type:

Biochemical

Assay Sub Type:

Enzymatic

Functional Mode:

Antagonist

Measured Response:

Scintillation

Testing Information

Tracer:

33P

ATP Concentration:

45 µM

Incubation:

40 min at RT

Test Sample Requirements:

Minimum for 1) Screen: 60 µl of 10 mM stock -OR- 1 mg (pre-weighed) for 10µM final testing. 2) Dose Response: 90 µl of 10 mM stock -OR- 1 mg (pre-weighed) for a top concentration at 10 µM.

Minimum Order Quantity:

10

Turnaround Time

Standard:

15 Business Days

Reference Compound Data

PubChem ID

122130844

Name

Staurosporine

Measurement

0.154nM - IC50

Clinical Relevance

Therapeutic Area:

Oncology/Immuno-Oncology

Additional Information

Brand:

LeadHunter

Testing Location:

France - Celle L'Evescault