OVERVIEW
DOCUMENTS/REFERENCES
Biological Information
No. of Assays on Panel:
95
Assays on Panel:
Family
GPCR
Name
NK1 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
100
Protein
NK1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2C Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1003
Protein
5-HT2C
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NK2 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
102
Protein
NK2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NK3 Human Tachykinin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
104
Protein
NK3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Neuropeptide Y (Non-Selective) Rat GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
105
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
alpha2 (Non-Selective) Rat Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
11
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Lipid Metabolism
Name
COX1 Human Cyclooxygenase Enzymatic LeadHunter Assay - TW
Item
116030
Protein
COX1
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
B1 Human Bradykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1189
Protein
B1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H2 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1208
Protein
H2
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (Non-Selective) Rat Ion Channel [3H] TCP Binding LeadHunter Assay - FR
Item
124
Protein
NMDA(PCP site)
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
131
Protein
5-HT1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H3 Human Histamine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1332
Protein
H3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CRF1 Human Corticotropin-Releasing Factor GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1467
Protein
CRF1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MT1 Human Melatonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1538
Protein
MT1
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
CHT1 Human Choline Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1552
Protein
CHT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
V1A Human Vasopressin / Oxytocin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
159
Protein
V1A
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Rat Calcium Ion Channel Binding (Verapamil Site) LeadHunter Assay - FR
Item
163
Protein
CaV1.2 (Vera. site)
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
KV (Non-Selective) Rat Potassium Ion Channel [125I] alpha-Dendrotoxin Binding LeadHunter Assay - FR
Item
166
Protein
Kv1.1
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
SKCa (Non-Selective) Rat Potassium Ion Channel [125I] Apamin Binding LeadHunter Assay - FR
Item
167
Protein
SKCa
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
beta1 Human Adrenoceptor GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
18
Protein
beta1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
EP2 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1955
Protein
EP2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A1 Human Adenosine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
2
Protein
A1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta2 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
20
Protein
beta2
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
ATPase (Na+/K+) Pig Brain Enzymatic LeadHunter Assay - FR
Item
2009
Protein
Na/K ATPase
Organism
Pig
Assay Sub Type
Enzymatic
Family
PDE
Name
PDE5 (Non-Selective) Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
204
Protein
PDE5
Organism
Human
Assay Sub Type
Enzymatic
Family
Epigenetic
Name
HDAC3 Human Histone Deacetylase (HDAC) Enzymatic LeadHunter Assay - FR
Item
2083
Protein
HDAC3
Organism
Human
Assay Sub Type
Enzymatic
Family
Neurotransmitter Metabolism
Name
Tyrosine Hydroxylase Rat Enzymatic LeadHunter Assay - FR
Item
214
Protein
Tyrosine Hydroxylase
Organism
Rat
Assay Sub Type
Enzymatic
Family
DNA Repair & Mitotic Regulation
Name
CENPE Human PPP1R Enzymatic LeadHunter Assay - FR
Item
2150
Protein
CENPE
Organism
Human
Assay Sub Type
Enzymatic
Family
DNA Repair & Mitotic Regulation
Name
EG5 Human Kinesin Enzymatic LeadHunter Assay - FR
Item
2151
Protein
EG5
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
IP Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
2230
Protein
IP
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
PR Human Progesterone NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
2341
Protein
PR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
AT1 Human Angiotensin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
24
Protein
AT1
Organism
Human
Assay Sub Type
Binding
Family
Epigenetic
Name
HDAC4 Human Histone Deacetylase (HDAC) Enzymatic LeadHunter Assay - FR
Item
2493
Protein
HDAC4
Organism
Human
Assay Sub Type
Enzymatic
Family
Epigenetic
Name
HDAC6 Human Histone Deacetylase (HDAC) Enzymatic LeadHunter Assay - FR
Item
2495
Protein
HDAC6
Organism
Human
Assay Sub Type
Enzymatic
Family
Epigenetic
Name
Sirtuin 1 Human Histone Deacetylase (HDAC) Enzymatic Antagonist LeadHunter Assay - FR
Item
2581
Protein
Sirtuin 1
Organism
Human
Assay Sub Type
Enzymatic
Family
Epigenetic
Name
Sirtuin 2 Human Histone Deacetylase (HDAC) Enzymatic Antagonist LeadHunter Assay - FR
Item
2582
Protein
Sirtuin 2
Organism
Human
Assay Sub Type
Enzymatic
Family
Phosphatase
Name
PTP1B Human Phosphatase Enzymatic LeadHunter Assay - FR
Item
2593
Protein
PTP1B
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
AT2 Human Angiotensin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
26
Protein
AT2
Organism
Human
Assay Sub Type
Binding
Family
Epigenetic
Name
HDAC11 Human Histone Deacetylase (HDAC) Enzymatic LeadHunter Assay - FR
Item
2663
Protein
HDAC11
Organism
Human
Assay Sub Type
Enzymatic
Family
Nucleotide Signaling
Name
Adenylyl Cyclase Hamster Enzymatic Agonist LeadHunter Assay - FR
Item
3002
Protein
Organism
Hamster
Assay Sub Type
Enzymatic
Family
Ion Channel
Name
nAChR (alpha4/beta2) Human Ion Channel Binding Agonist Radioligand LeadHunter Assay - FR
Item
3029
Protein
nAChR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
B2 Human Bradykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
33
Protein
B2
Organism
Human
Assay Sub Type
Binding
Family
Enzyme
Name
Monoamine Oxidase B (MAO-B) Human Enzymatic LeadHunter Assay - FR
Item
3477
Protein
MAO-B
Organism
Human
Assay Sub Type
Enzymatic
Family
Transmembrane (Other)
Name
sigma (Non-Selective) Human Binding Agonist Radioligand LeadHunter Assay - FR
Item
3500
Protein
Sigma1/Sigma2
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
NET Human Norepinephrine Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
355
Protein
NET
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NOP (ORL1) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
358
Protein
NOP (ORL1)
Organism
Human
Assay Sub Type
Binding
Family
Enzyme
Name
Acetylcholinesterase Human Enzymatic LeadHunter Assay - FR
Item
363
Protein
AChE
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
CB2 Human Cannabinoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
37
Protein
CB2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CCK1 (CCKA) Human Cholecystokinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
39
Protein
CCK1 (CCKA)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A2A Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4
Protein
A2A
Organism
Human
Assay Sub Type
Binding
Family
PDE
Name
PDE1B Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
4070
Protein
PDE1B
Organism
Human
Assay Sub Type
Enzymatic
Family
PDE
Name
PDE2A1 Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
4071
Protein
PDE2A
Organism
Human
Assay Sub Type
Enzymatic
Family
Enzyme
Name
PDE3A Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
4072
Protein
PDE3A
Organism
Human
Assay Sub Type
Enzymatic
Family
Enzyme
Name
PDE4D2 Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
4077
Protein
PDE4D
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
CCK2 (CCKB) Human Cholecystokinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
41
Protein
CCK2 (CCKB)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MC4 Human Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
420
Protein
MC4
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
SERT Human Serotonin Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
439
Protein
SERT
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D1 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
44
Protein
D1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (alpha1/beta2/gamma2) Human Ion Channel [3H] Flunitrazepam Binding Agonist Radioligand LeadHunter Assay - FR
Item
4518
Protein
GABAA(BZD site)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (diltiazem site) (benzothiazepines) LeadHunter Assay - FR
Item
4549
Protein
Cav1.2 (L-type)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D2S Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
46
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
Neurotransmitter Metabolism
Name
GABA Transaminase Rat Enzymatic LeadHunter Assay - FR
Item
461
Protein
GABA Transaminase
Organism
Rat
Assay Sub Type
Enzymatic
Family
NHR
Name
GR Human Glucocorticoid NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
469
Protein
GR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CB1 Human Cannabinoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4708
Protein
CB1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
471
Protein
5-HT2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D3 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
48
Protein
D3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D4.4 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
49
Protein
D4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
V2 Human Vasopressin / Oxytocin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
497
Protein
V2
Organism
Human
Assay Sub Type
Binding
Family
Enzyme
Name
Monoamine Oxidase A (MAO-A) Human Enzymatic LeadHunter Assay - FR
Item
5108
Protein
MAO-A
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
Non-Selective Rat Opioid GPCR Mass Spectrometry Binding Antagonist Ligand LeadHunter Assay - FR
Item
5110
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
KATP Rat Potassium Ion Channel Mass Spectrometry Binding Antagonist Ligand LeadHunter Assay - FR
Item
5111
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Transmembrane (Other)
Name
Imidazoline I2 Rat Mass Spectrometry Binding Antagonist Ligand LeadHunter Assay - FR
Item
5114
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Transporter
Name
DAT Human Dopamine Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
52
Protein
DAT
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GluK2 Human Ion Channel [3H] Kainic acid Binding LeadHunter Assay - FR
Item
5379
Protein
Kainate
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
ETA Human Endothelin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
54
Protein
ETA
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
ERalpha Human Estrogen NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
5484
Protein
ERalpha
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (Dihydropyridine Site) LeadHunter Assay - FR
Item
5538
Protein
CaV1.2 (DHP site)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Sodium Channel Site2 (Non-selective) Rat Ion Channel Batrachotoxin Mass Spectrometry Binding LeadHunter Assay - FR
Item
5572
Protein
Nav1.5
Organism
Rat
Assay Sub Type
Binding
Family
Phosphatase
Name
CDC25A Human Phosphatase Enzymatic LeadHunter Assay - FR
Item
5598
Protein
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
ETB Human Endothelin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
56
Protein
ETB
Organism
Human
Assay Sub Type
Binding
Family
Kinase
Name
PKCalpha Human PKC Kinase Enzymatic Radiometric [Km ATP] SafetyScreen - FR
Item
5625
Protein
PKCalpha
Organism
Human
Assay Sub Type
Enzymatic
Family
Ion Channel
Name
GABAA (alpha1/beta2/gamma2) Human Ion Channel Picrotoxinin Mass Spectrometry Binding Antagonist Ligand LeadHunter Assay - FR
Item
5666
Protein
GABAA
Organism
Human
Assay Sub Type
Binding
Family
Other
Name
GABA (Non-Selective) Rat Receptors [3H] GABA Binding Agonist Radioligand LeadHunter Assay - FR
Item
57
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Transporter
Name
GAT1 Human GABA Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
5773
Protein
GAT-1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CysLT1 Human Leukotriene GPCR Mass Spectrometry Binding Agonist ligand LeadHunter Assay - FR
Item
5841
Protein
CYSLT1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (NMDA, NR1/NR2A) Human Ion Channel [3H] CGP-39653 Binding LeadHunter Assay - FR
Item
5875
Protein
GluN1 / GluN2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A3 Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
6
Protein
A3
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (AMPA, Non-Selective) Rat Ion Channel [3H] AMPA Binding LeadHunter Assay - FR
Item
64
Protein
AMPA
Organism
Rat
Assay Sub Type
Binding
Family
NHR
Name
PPARgamma Human NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
641
Protein
PPARgamma
Organism
Human
Assay Sub Type
Binding
Family
Lipid Metabolism
Name
5-LOX Human Lipoxygenase Enzymatic LeadHunter Assay - FR
Item
772
Protein
5-LOX
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
alpha1 (Non-Selective) Rat Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
8
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
H1 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
870
Protein
H1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Acetylcholine (Muscarinic, Non-Selective) Rat GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
89
Protein
Organism
Rat
Assay Sub Type
Binding
Family
NHR
Name
AR Human Androgen NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
933
Protein
AR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
P2Y (Non-Selective) Rat GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
EU-6000
Protein
Organism
Rat
Assay Sub Type
Binding
Testing Information
Test Sample Requirements:
Minimum for Screen: 180 µl of 10 mM stock -OR- 1 mg (pre-weighed) for 10µM final testing.
(PBS or HBSS working solutions are not compatible)
Turnaround Time
Standard:
15 Business Days
Additional Information
Brand:
LeadHunter
Testing Location:
France - Celle L'Evescault
Questions? Contact Us
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