OVERVIEW
DOCUMENTS/REFERENCES
Biological Information
No. of Assays on Panel:
79
Assays on Panel:
Family
GPCR
Name
NK1 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
100
Protein
NK1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NK2 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
102
Protein
NK2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NK3 Human Tachykinin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
104
Protein
NK3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Y1 Human Neuropeptide Y GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
106
Protein
Y1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Y2 Human Neuropeptide Y GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
107
Protein
Y2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NT1 Human Neurotensin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
109
Protein
NT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha2 (Non-Selective) Rat Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
11
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
delta (DOP) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
114
Protein
delta (DOP)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
mu (MOP) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
118
Protein
mu (MOP)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H2 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1208
Protein
H2
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (Non-Selective) Rat Ion Channel [3H] TCP Binding LeadHunter Assay - FR
Item
124
Protein
NMDA(PCP site)
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
131
Protein
5-HT1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2B Human Serotonin GPCR [125I](±)DOI Binding Agonist Radioligand LeadHunter Assay - FR
Item
1333
Protein
5-HT2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2A Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
135
Protein
5-HT2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2C Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
137
Protein
5-HT2C
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT5A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
140
Protein
5-HT5A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT6 Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
142
Protein
5-HT6
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT7 Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
144
Protein
5-HT7
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Somatostatin (Non-Selective) Mouse GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
149
Protein
Organism
Mouse
Assay Sub Type
Binding
Family
GPCR
Name
PAC1 (PACAP) Human VIP and PACAP GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1518
Protein
PAC1 (PACAP)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MT1 Human Melatonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1538
Protein
MT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
VIP1 (VPAC1) Human VIP and PACAP GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
157
Protein
VIP1 (VPAC1)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
V1A Human Vasopressin / Oxytocin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
159
Protein
V1A
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Rat Calcium Ion Channel Binding (Verapamil Site) LeadHunter Assay - FR
Item
163
Protein
CaV1.2 (Vera. site)
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
KV (Non-Selective) Rat Potassium Ion Channel [125I] alpha-Dendrotoxin Binding LeadHunter Assay - FR
Item
166
Protein
Kv1.1
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
SKCa (Non-Selective) Rat Potassium Ion Channel [125I] Apamin Binding LeadHunter Assay - FR
Item
167
Protein
SKCa
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
beta1 Human Adrenoceptor GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
18
Protein
beta1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
EP2 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1955
Protein
EP2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A1 Human Adenosine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
2
Protein
A1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta2 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
20
Protein
beta2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
IP Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
2230
Protein
IP
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
AT1 Human Angiotensin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
24
Protein
AT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
AT2 Human Angiotensin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
26
Protein
AT2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Bombesin (Non-Selective) Rat GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
30
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
B2 Human Bradykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
33
Protein
B2
Organism
Human
Assay Sub Type
Binding
Family
Transmembrane (Other)
Name
sigma (Non-Selective) Human Binding Agonist Radioligand LeadHunter Assay - FR
Item
3500
Protein
Sigma1/Sigma2
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
NET Human Norepinephrine Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
355
Protein
NET
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NOP (ORL1) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
358
Protein
NOP (ORL1)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CCR1 Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
361
Protein
CCR1
Organism
Human
Assay Sub Type
Binding
Family
Mitochondrial Function
Name
PBR Human Binding Antagonist Radioligand LeadHunter Assay - FR
Item
3643
Protein
PBR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CGRP (CLR/RAMP1) Human Calcitonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
373
Protein
CLR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CCK1 (CCKA) Human Cholecystokinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
39
Protein
CCK1 (CCKA)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A2A Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4
Protein
A2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CCK2 (CCKB) Human Cholecystokinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
41
Protein
CCK2 (CCKB)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
GAL2 Human Galanin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
410
Protein
GAL2
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
5-HT3 Human Serotonin Ion Channel Binding Antagonist Radioligand LeadHunter Assay - FR
Item
411
Protein
5-HT3A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CXCR2 (IL-8RB) Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
419
Protein
CXCR2 (IL-8RB)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MC4 Human Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
420
Protein
MC4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1B Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
4376
Protein
5-HT1B
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
SERT Human Serotonin Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
439
Protein
SERT
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D1 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
44
Protein
D1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
EP4 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
441
Protein
EP4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
kappa (KOP) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4461
Protein
kappa (KOP)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (alpha1/beta2/gamma2) Human Ion Channel [3H] Flunitrazepam Binding Agonist Radioligand LeadHunter Assay - FR
Item
4518
Protein
GABAA(BZD site)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D2S Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
46
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
GR Human Glucocorticoid NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
469
Protein
GR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CB1 Human Cannabinoid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4708
Protein
CB1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D3 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
48
Protein
D3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D4.4 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
49
Protein
D4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D5 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
50
Protein
D5
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
DAT Human Dopamine Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
52
Protein
DAT
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
ETA Human Endothelin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
54
Protein
ETA
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Sodium Channel Site2 (Non-selective) Rat Ion Channel Batrachotoxin Mass Spectrometry Binding LeadHunter Assay - FR
Item
5572
Protein
Nav1.5
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
ETB Human Endothelin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
56
Protein
ETB
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (alpha1/beta2/gamma2) Human Ion Channel Picrotoxinin Mass Spectrometry Binding Antagonist Ligand LeadHunter Assay - FR
Item
5666
Protein
GABAA
Organism
Human
Assay Sub Type
Binding
Family
Other
Name
GABA (Non-Selective) Rat Receptors [3H] GABA Binding Agonist Radioligand LeadHunter Assay - FR
Item
57
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
A3 Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
6
Protein
A3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
GAL1 Human Galanin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
62
Protein
GAL1
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
PPARgamma Human NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
641
Protein
PPARgamma
Organism
Human
Assay Sub Type
Binding
Family
Kinase
Name
PDGFR (Non-Selective) Mouse RTK Kinase Binding Agonist Radioligand LeadHunter Assay - FR
Item
70
Protein
Organism
Mouse
Assay Sub Type
Binding
Family
Cell Surface (Other)
Name
TNF-alpha Human Binding Agonist Radioligand LeadHunter Assay - FR
Item
76
Protein
TNF-alpha
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha1 (Non-Selective) Rat Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
8
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
H1 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
870
Protein
H1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M1 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
91
Protein
M1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M2 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
93
Protein
M2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M3 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
95
Protein
M3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M4 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
96
Protein
M4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M5 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
97
Protein
M5
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
P2Y (Non-Selective) Rat GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
EU-6000
Protein
Organism
Rat
Assay Sub Type
Binding
Testing Information
Test Sample Requirements:
Minimum for Screen: 130 μl of 10 mM stock -OR- 1 mg (pre-weighed) for 10µM final testing.
Turnaround Time
Standard:
10 Business Days
Additional Information
Brand:
LeadHunter
Testing Location:
France - Celle L'Evescault
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