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Matrix
Example Data Type:
Secondary Screen (Kd)
Primary Screen(% control or competition)
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Assay Data File:
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Bromodomain
Kd
Primary
To highlight spots, select a compound(s), click 'fill' and select entries.
Create Images for:
Crizotinib
Highlight These Spots (
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):
Crizotinib|SgK110|240
Crizotinib|SIK2|200
Crizotinib|SLK|18
Crizotinib|SNARK|120
Crizotinib|SRC|560
Crizotinib|SRPK1|1800
Crizotinib|SRPK3|8200
Crizotinib|STK35|610
Crizotinib|SYK|2500
Crizotinib|TAK1|1800
Crizotinib|TAOK1|1200
Crizotinib|TAOK2|900
Crizotinib|TAOK3|490
Crizotinib|TBK1|690
Crizotinib|TESK1|380
Crizotinib|TGFBR1|1000
Crizotinib|TIE1|110
Crizotinib|TIE2|270
Crizotinib|TNK1|320
Crizotinib|TNK2|760
Crizotinib|TNNI3K|110
Crizotinib|TRKA|95
Crizotinib|TRKB|37
Crizotinib|TRKC|82
Crizotinib|TXK|850
Crizotinib|TYK2(JH1domain-catalytic)|210
Crizotinib|TYK2(JH2domain-pseudokinase)|2000
Crizotinib|TYRO3|800
Crizotinib|ULK1|1000
Crizotinib|ULK2|1600
Crizotinib|ULK3|6700
Crizotinib|YES|770
Crizotinib|YSK4|980
Crizotinib|ZAP70|4200
Crizotinib|AAK1|2300
Crizotinib|ABL1-nonphosphorylated|78
Crizotinib|ABL2|460
Crizotinib|ACVR1|440
Crizotinib|ACVR1B|860
Crizotinib|ADCK4|1100
Crizotinib|ALK|3.3
Crizotinib|AMPK-alpha1|2400
Crizotinib|ANKK1|780
Crizotinib|AURKA|260
Crizotinib|AURKB|76
Crizotinib|AURKC|4300
Crizotinib|AXL|7.8
Crizotinib|BIKE|740
Crizotinib|BLK|110
Crizotinib|BMPR1B|230
Crizotinib|BMX|3600
Crizotinib|BTK|7800
Crizotinib|CAMKK2|1500
Crizotinib|CASK|140
Crizotinib|CDC2L1|760
Crizotinib|CDC2L2|420
Crizotinib|CDK7|330
Crizotinib|CDKL2|2100
Crizotinib|CSF1R|210
Crizotinib|DCAMKL1|330
Crizotinib|DCAMKL2|370
Crizotinib|DDR1|510
Crizotinib|DLK|170
Crizotinib|DMPK|1400
Crizotinib|DYRK2|4000
Crizotinib|EPHA1|140
Crizotinib|EPHA2|100
Crizotinib|EPHA3|700
Crizotinib|EPHA4|360
Crizotinib|EPHA5|1000
Crizotinib|EPHA6|65
Crizotinib|EPHA7|470
Crizotinib|EPHA8|280
Crizotinib|EPHB1|120
Crizotinib|EPHB4|570
Crizotinib|EPHB6|6
Crizotinib|ERK5|510
Crizotinib|FAK|310
Crizotinib|FER|270
Crizotinib|FES|450
Crizotinib|FGFR3|2700
Crizotinib|FGR|670
Crizotinib|FLT1|2300
Crizotinib|FLT3|850
Crizotinib|FRK|2900
Crizotinib|FYN|1300
Crizotinib|GRK4|4200
Crizotinib|HIPK4|3600
Crizotinib|HPK1|39
Crizotinib|IGF1R|780
Crizotinib|IKK-beta|5500
Crizotinib|IKK-epsilon|710
Crizotinib|INSR|340
Crizotinib|INSRR|600
Crizotinib|IRAK1|49
Crizotinib|IRAK3|31
Crizotinib|IRAK4|3600
Crizotinib|ITK|2000
Crizotinib|JAK1(JH1domain-catalytic)|330
Crizotinib|JAK2(JH1domain-catalytic)|290
Crizotinib|JAK3(JH1domain-catalytic)|200
Crizotinib|LCK|30
Crizotinib|LIMK1|830
Crizotinib|LIMK2|690
Crizotinib|LOK|44
Crizotinib|LTK|12
Crizotinib|LYN|940
Crizotinib|LZK|230
Crizotinib|MAP3K1|1100
Crizotinib|MAP3K15|2800
Crizotinib|MAP3K2|72
Crizotinib|MAP3K3|110
Crizotinib|MAP4K2|80
Crizotinib|MAP4K3|75
Crizotinib|MAP4K5|79
Crizotinib|MEK3|3300
Crizotinib|MERTK|3.6
Crizotinib|MET|2.1
Crizotinib|MINK|4400
Crizotinib|MST1|580
Crizotinib|MST1R|25
Crizotinib|MST2|990
Crizotinib|MST4|2800
Crizotinib|MUSK|230
Crizotinib|NEK7|5700
Crizotinib|NEK9|790
Crizotinib|NIM1|4600
Crizotinib|PIP5K1A|3200
Crizotinib|PLK4|60
Crizotinib|PRKD1|990
Crizotinib|PRKD3|510
Crizotinib|PRKR|1100
Crizotinib|PYK2|190
Crizotinib|RIOK1|6100
Crizotinib|RIOK3|4000
Crizotinib|RIPK1|1600
Crizotinib|RIPK2|900
Crizotinib|RIPK4|2100
Crizotinib|RIPK5|450
Crizotinib|ROCK1|3700
Crizotinib|ROCK2|3300
Crizotinib|ROS1|4.1
Crizotinib|S6K1|640
Crizotinib|SBK1|1300
Crizotinib|SgK110
Crizotinib|SIK2
Crizotinib|SLK
Crizotinib|SNARK
Crizotinib|SRC
Crizotinib|SRPK1
Crizotinib|SRPK3
Crizotinib|STK35
Crizotinib|SYK
Crizotinib|TAK1
Crizotinib|TAOK1
Crizotinib|TAOK2
Crizotinib|TAOK3
Crizotinib|TBK1
Crizotinib|TESK1
Crizotinib|TGFBR1
Crizotinib|TIE1
Crizotinib|TIE2
Crizotinib|TNK1
Crizotinib|TNK2
Crizotinib|TNNI3K
Crizotinib|TRKA
Crizotinib|TRKB
Crizotinib|TRKC
Crizotinib|TXK
Crizotinib|TYK2(JH1domain-catalytic)
Crizotinib|TYK2(JH2domain-pseudokinase)
Crizotinib|TYRO3
Crizotinib|ULK1
Crizotinib|ULK2
Crizotinib|ULK3
Crizotinib|YES
Crizotinib|YSK4
Crizotinib|ZAP70
Crizotinib|AAK1
Crizotinib|ABL1-nonphosphorylated
Crizotinib|ABL2
Crizotinib|ACVR1
Crizotinib|ACVR1B
Crizotinib|ADCK4
Crizotinib|ALK
Crizotinib|AMPK-alpha1
Crizotinib|ANKK1
Crizotinib|AURKA
Crizotinib|AURKB
Crizotinib|AURKC
Crizotinib|AXL
Crizotinib|BIKE
Crizotinib|BLK
Crizotinib|BMPR1B
Crizotinib|BMX
Crizotinib|BTK
Crizotinib|CAMKK2
Crizotinib|CASK
Crizotinib|CDC2L1
Crizotinib|CDC2L2
Crizotinib|CDK7
Crizotinib|CDKL2
Crizotinib|CSF1R
Crizotinib|DCAMKL1
Crizotinib|DCAMKL2
Crizotinib|DDR1
Crizotinib|DLK
Crizotinib|DMPK
Crizotinib|DYRK2
Crizotinib|EPHA1
Crizotinib|EPHA2
Crizotinib|EPHA3
Crizotinib|EPHA4
Crizotinib|EPHA5
Crizotinib|EPHA6
Crizotinib|EPHA7
Crizotinib|EPHA8
Crizotinib|EPHB1
Crizotinib|EPHB4
Crizotinib|EPHB6
Crizotinib|ERK5
Crizotinib|FAK
Crizotinib|FER
Crizotinib|FES
Crizotinib|FGFR3
Crizotinib|FGR
Crizotinib|FLT1
Crizotinib|FLT3
Crizotinib|FRK
Crizotinib|FYN
Crizotinib|GRK4
Crizotinib|HIPK4
Crizotinib|HPK1
Crizotinib|IGF1R
Crizotinib|IKK-beta
Crizotinib|IKK-epsilon
Crizotinib|INSR
Crizotinib|INSRR
Crizotinib|IRAK1
Crizotinib|IRAK3
Crizotinib|IRAK4
Crizotinib|ITK
Crizotinib|JAK1(JH1domain-catalytic)
Crizotinib|JAK2(JH1domain-catalytic)
Crizotinib|JAK3(JH1domain-catalytic)
Crizotinib|LCK
Crizotinib|LIMK1
Crizotinib|LIMK2
Crizotinib|LOK
Crizotinib|LTK
Crizotinib|LYN
Crizotinib|LZK
Crizotinib|MAP3K1
Crizotinib|MAP3K15
Crizotinib|MAP3K2
Crizotinib|MAP3K3
Crizotinib|MAP4K2
Crizotinib|MAP4K3
Crizotinib|MAP4K5
Crizotinib|MEK3
Crizotinib|MERTK
Crizotinib|MET
Crizotinib|MINK
Crizotinib|MST1
Crizotinib|MST1R
Crizotinib|MST2
Crizotinib|MST4
Crizotinib|MUSK
Crizotinib|NEK7
Crizotinib|NEK9
Crizotinib|NIM1
Crizotinib|PIP5K1A
Crizotinib|PLK4
Crizotinib|PRKD1
Crizotinib|PRKD3
Crizotinib|PRKR
Crizotinib|PYK2
Crizotinib|RIOK1
Crizotinib|RIOK3
Crizotinib|RIPK1
Crizotinib|RIPK2
Crizotinib|RIPK4
Crizotinib|RIPK5
Crizotinib|ROCK1
Crizotinib|ROCK2
Crizotinib|ROS1
Crizotinib|S6K1
Crizotinib|SBK1
Crizotinib|SgK110|240
Crizotinib|SIK2|200
Crizotinib|SLK|18
Crizotinib|SNARK|120
Crizotinib|SRC|560
Crizotinib|SRPK1|1800
Crizotinib|SRPK3|8200
Crizotinib|STK35|610
Crizotinib|SYK|2500
Crizotinib|TAK1|1800
Crizotinib|TAOK1|1200
Crizotinib|TAOK2|900
Crizotinib|TAOK3|490
Crizotinib|TBK1|690
Crizotinib|TESK1|380
Crizotinib|TGFBR1|1000
Crizotinib|TIE1|110
Crizotinib|TIE2|270
Crizotinib|TNK1|320
Crizotinib|TNK2|760
Crizotinib|TNNI3K|110
Crizotinib|TRKA|95
Crizotinib|TRKB|37
Crizotinib|TRKC|82
Crizotinib|TXK|850
Crizotinib|TYK2(JH1domain-catalytic)|210
Crizotinib|TYK2(JH2domain-pseudokinase)|2000
Crizotinib|TYRO3|800
Crizotinib|ULK1|1000
Crizotinib|ULK2|1600
Crizotinib|ULK3|6700
Crizotinib|YES|770
Crizotinib|YSK4|980
Crizotinib|ZAP70|4200
Crizotinib|AAK1|2300
Crizotinib|ABL1-nonphosphorylated|78
Crizotinib|ABL2|460
Crizotinib|ACVR1|440
Crizotinib|ACVR1B|860
Crizotinib|ADCK4|1100
Crizotinib|ALK|3.3
Crizotinib|AMPK-alpha1|2400
Crizotinib|ANKK1|780
Crizotinib|AURKA|260
Crizotinib|AURKB|76
Crizotinib|AURKC|4300
Crizotinib|AXL|7.8
Crizotinib|BIKE|740
Crizotinib|BLK|110
Crizotinib|BMPR1B|230
Crizotinib|BMX|3600
Crizotinib|BTK|7800
Crizotinib|CAMKK2|1500
Crizotinib|CASK|140
Crizotinib|CDC2L1|760
Crizotinib|CDC2L2|420
Crizotinib|CDK7|330
Crizotinib|CDKL2|2100
Crizotinib|CSF1R|210
Crizotinib|DCAMKL1|330
Crizotinib|DCAMKL2|370
Crizotinib|DDR1|510
Crizotinib|DLK|170
Crizotinib|DMPK|1400
Crizotinib|DYRK2|4000
Crizotinib|EPHA1|140
Crizotinib|EPHA2|100
Crizotinib|EPHA3|700
Crizotinib|EPHA4|360
Crizotinib|EPHA5|1000
Crizotinib|EPHA6|65
Crizotinib|EPHA7|470
Crizotinib|EPHA8|280
Crizotinib|EPHB1|120
Crizotinib|EPHB4|570
Crizotinib|EPHB6|6
Crizotinib|ERK5|510
Crizotinib|FAK|310
Crizotinib|FER|270
Crizotinib|FES|450
Crizotinib|FGFR3|2700
Crizotinib|FGR|670
Crizotinib|FLT1|2300
Crizotinib|FLT3|850
Crizotinib|FRK|2900
Crizotinib|FYN|1300
Crizotinib|GRK4|4200
Crizotinib|HIPK4|3600
Crizotinib|HPK1|39
Crizotinib|IGF1R|780
Crizotinib|IKK-beta|5500
Crizotinib|IKK-epsilon|710
Crizotinib|INSR|340
Crizotinib|INSRR|600
Crizotinib|IRAK1|49
Crizotinib|IRAK3|31
Crizotinib|IRAK4|3600
Crizotinib|ITK|2000
Crizotinib|JAK1(JH1domain-catalytic)|330
Crizotinib|JAK2(JH1domain-catalytic)|290
Crizotinib|JAK3(JH1domain-catalytic)|200
Crizotinib|LCK|30
Crizotinib|LIMK1|830
Crizotinib|LIMK2|690
Crizotinib|LOK|44
Crizotinib|LTK|12
Crizotinib|LYN|940
Crizotinib|LZK|230
Crizotinib|MAP3K1|1100
Crizotinib|MAP3K15|2800
Crizotinib|MAP3K2|72
Crizotinib|MAP3K3|110
Crizotinib|MAP4K2|80
Crizotinib|MAP4K3|75
Crizotinib|MAP4K5|79
Crizotinib|MEK3|3300
Crizotinib|MERTK|3.6
Crizotinib|MET|2.1
Crizotinib|MINK|4400
Crizotinib|MST1|580
Crizotinib|MST1R|25
Crizotinib|MST2|990
Crizotinib|MST4|2800
Crizotinib|MUSK|230
Crizotinib|NEK7|5700
Crizotinib|NEK9|790
Crizotinib|NIM1|4600
Crizotinib|PIP5K1A|3200
Crizotinib|PLK4|60
Crizotinib|PRKD1|990
Crizotinib|PRKD3|510
Crizotinib|PRKR|1100
Crizotinib|PYK2|190
Crizotinib|RIOK1|6100
Crizotinib|RIOK3|4000
Crizotinib|RIPK1|1600
Crizotinib|RIPK2|900
Crizotinib|RIPK4|2100
Crizotinib|RIPK5|450
Crizotinib|ROCK1|3700
Crizotinib|ROCK2|3300
Crizotinib|ROS1|4.1
Crizotinib|S6K1|640
Crizotinib|SBK1|1300
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Crizotinib
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Crizotinib
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* WildType kinase assays appear in both the main TREEspot and Mutant kinase dendrogams.
Human Kinome image created by KINOMEscan.
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Crizotinib
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SgK110
SIK2
SLK
SNARK
SRC
SRPK1
STK35
SYK
TAK1
TAOK1
TAOK2
TAOK3
TBK1
TESK1
TGFBR1
TIE1
TIE2
TNK1
TNK2
TNNI3K
TRKA
TRKB
TRKC
TXK
TYK2(JH1domain-catalytic)
TYK2(JH2domain-pseudokinase)
TYRO3
ULK1
ULK2
YES
YSK4
AAK1
ABL1-nonphosphorylated
ABL1-nonphosphorylated
ABL2
ACVR1
ACVR1B
ADCK4
ALK
ALK
AMPK-alpha1
ANKK1
AURKA
AURKB
AXL
BIKE
BLK
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CAMKK2
CASK
CDC2L1
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CDKL2
CSF1R
DCAMKL1
DCAMKL2
DDR1
DLK
DMPK
EPHA1
EPHA2
EPHA3
EPHA4
EPHA5
EPHA6
EPHA7
EPHA8
EPHB1
EPHB4
EPHB6
ERK5
FAK
FER
FES
FGFR3
FGFR3
FGR
FLT1
FLT3
FLT3
FRK
FYN
HPK1
IGF1R
IKK-epsilon
INSR
INSRR
IRAK1
IRAK3
ITK
JAK1(JH1domain-catalytic)
JAK2(JH1domain-catalytic)
JAK3(JH1domain-catalytic)
LCK
LIMK1
LIMK2
LOK
LTK
LYN
LZK
MAP3K1
MAP3K15
MAP3K2
MAP3K3
MAP4K2
MAP4K3
MAP4K5
MERTK
MET
MET
MST1
MST1R
MST2
MST4
MUSK
NEK9
PLK4
PRKD1
PRKD3
PRKR
PYK2
RIPK1
RIPK2
RIPK4
RIPK5
ROS1
S6K1
SBK1
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